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Justina Kazokaitė-Adomaitienė
Justina Kazokaitė-Adomaitienė
The Netherlands Cancer Institute, Amsterdam
E-mail confirmado em nki.nl
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Benzenesulfonamides with pyrimidine moiety as inhibitors of human carbonic anhydrases I, II, VI, VII, XII, and XIII
E Čapkauskaitė, A Zubrienė, A Smirnov, J Torresan, M Kišonaitė, ...
Bioorganic & medicinal chemistry 21 (22), 6937-6947, 2013
512013
Functionalization of fluorinated benzenesulfonamides and their inhibitory properties toward carbonic anhydrases
V Dudutienė, A Zubrienė, A Smirnov, DD Timm, J Smirnovienė, ...
ChemMedChem 10 (4), 662-687, 2015
432015
4-Amino-substituted Benzenesulfonamides as Inhibitors of Human Carbonic Anhydrases
K Rutkauskas, A Zubrienė, I Tumosienė, K Kantminienė, M Kažemėkaitė, ...
Molecules 19 (11), 17356-17380, 2014
302014
Novel fluorinated carbonic anhydrase IX inhibitors reduce hypoxia-induced acidification and clonogenic survival of cancer cells
J Kazokaitė, R Niemans, V Dudutienė, HM Becker, J Leitāns, A Zubrienė, ...
Oncotarget 9 (42), 26800, 2018
252018
An update on anticancer drug development and delivery targeting carbonic anhydrase IX
J Kazokaitė, A Aspatwar, S Parkkila, D Matulis
PeerJ 5, e4068, 2017
252017
Intrinsic binding of 4‐substituted‐2, 3, 5, 6‐tetrafluorobenezenesulfonamides to native and recombinant human carbonic anhydrase VI
J Kazokaitė, G Milinavičiūtė, J Smirnovienė, J Matulienė, D Matulis
The FEBS Journal 282 (5), 972-983, 2015
222015
Fluorinated benzenesulfonamide anticancer inhibitors of carbonic anhydrase IX exhibit lower toxic effects on zebrafish embryonic development than ethoxzolamide
J Kazokaitė, A Aspatwar, V Kairys, S Parkkila, D Matulis
Drug and Chemical Toxicology 40 (3), 309-319, 2017
172017
Selective inhibition of human carbonic anhydrase IX in Xenopus oocytes and MDA-MB-231 breast cancer cells
J Kazokaitė, S Ames, HM Becker, JW Deitmer, D Matulis
Journal of Enzyme Inhibition and Medicinal Chemistry 31 (sup4), 38-44, 2016
122016
Actin maturation requires the ACTMAP/C19orf54 protease
P Haahr, RA Galli, LG van den Hengel, OB Bleijerveld, ...
Science 377 (6614), 1533-1537, 2022
102022
Engineered carbonic anhydrase VI-mimic enzyme switched the structure and affinities of inhibitors
J Kazokaitė, V Kairys, J Smirnovienė, A Smirnov, E Manakova, ...
Scientific reports 9 (1), 12710, 2019
42019
Engineering of chimeric carbonic anhydrases for designing isoform-selective inhibitors
J Smirnoviene, A Smirnov, V Kairys, J Kazokaite-Adomaitiene, ...
EUROPEAN BIOPHYSICS JOURNAL WITH BIOPHYSICS LETTERS 50 (SUPPL 1), 127-127, 2021
2021
Experimental approaches to identify selective picomolar inhibitors for carbonic anhydrase IX
J Kazokaitė-Adomaitienė, HM Becker, J Smirnovienė, LJ Dubois, ...
Current medicinal chemistry 28 (17), 3361-3384, 2021
2021
Development of fluorinated benzenesulfonamides as carbonic anhydrase IX inhibitors
V Dudutienė, A Zubrienė, J Kazokaitė, D Matulis
Chemistry and chemical technology: Lithuanian chemists conference, 2019 May …, 2019
2019
Efficacy of Novel CA IX Inhibitors in Biological Models
J Kazokaitė, HM Becker, HR Barker, A Aspatwar, S Parkkila, LJ Dubois, ...
Carbonic Anhydrase as Drug Target: Thermodynamics and Structure of Inhibitor …, 2019
2019
Investigation of human carbonic anhydrase VI and IX inhibitor efficacy and toxicity
J Kazokaitė
Vilniaus universitetas, 2018
2018
Discovery and Biological Characterization of Novel Selective Inhibitors of Carbonic Anhydrase IX
V Dudutienė, J Matulienė, A Smirnov, A Zubrienė, L Baranauskienė, ...
XIVth International conference of the Lithuanian biochemical society: the …, 2016
2016
Thermodynamics of anticancer drug lead binding to target proteins by thermal shift assay
A Zubrienė, J Gylytė, V Morkūnaitė, E Kazlauskas, L Baranauskienė, ...
Epigenetics–Bench to Bedside. COST Action TD0905: Program and Abstract Book …, 2013
2013
Thiophene sulfonamides as carbonic anhydrase inhibitors by titration calorimetry and thermal shift assay
V Morkūnaitė, A Zubrienė, L Baranauskienė, V Petrikaitė, J Gylytė, ...
Epigenetics: Bench to Bedside. COST Action TD0905: Abstract Book: April 26 …, 2012
2012
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