| Geometrically and conformationally restrained cinnamoyl compounds as inhibitors of HIV-1 integrase: synthesis, biological evaluation, and molecular modeling M Artico, R Di Santo, R Costi, E Novellino, G Greco, S Massa, ... Journal of medicinal chemistry 41 (21), 3948-3960, 1998 | 238 | 1998 |
| 5-Alkyl-2-(alkylthio)-6-(2,6-dihalophenylmethyl)-3,4-dihydropyrimidin-4(3H)-ones: Novel Potent and Selective Dihydro-alkoxy-benzyl-oxopyrimidine Derivatives A Mai, M Artico, G Sbardella, S Massa, E Novellino, G Greco, AG Loi, ... Journal of Medicinal Chemistry 42 (4), 619-627, 1999 | 159 | 1999 |
| Structure-based design, synthesis, and biological evaluation of novel pyrrolyl aryl sulfones: HIV-1 non-nucleoside reverse transcriptase inhibitors active at nanomolar … M Artico, R Silvestri, E Pagnozzi, B Bruno, E Novellino, G Greco, S Massa, ... Journal of Medicinal Chemistry 43 (9), 1886-1891, 2000 | 148 | 2000 |
| Pyrroloquinoxaline Derivatives as High-Affinity and Selective 5-HT3 Receptor Agonists: Synthesis, Further Structure−Activity Relationships, and Biological Studies G Campiani, E Morelli, S Gemma, V Nacci, S Butini, M Hamon, ... Journal of medicinal chemistry 42 (21), 4362-4379, 1999 | 138 | 1999 |
| Structure-based design, synthesis, and biological evaluation of conformationally restricted novel 2-alkylthio-6-[1-(2, 6-difluorophenyl) alkyl]-3, 4-dihydro-5-alkylpyrimidin-4 … A Mai, G Sbardella, M Artico, R Ragno, S Massa, E Novellino, G Greco, ... Journal of medicinal chemistry 44 (16), 2544-2554, 2001 | 136 | 2001 |
| A critical review of recent CoMFA applications KH Kim, G Greco, E Novellino Perspectives in drug discovery and design 12 (14), 257-315, 1998 | 126 | 1998 |
| Quinoxalinylethylpyridylthioureas (QXPTs) as potent non-nucleoside HIV-1 reverse transcriptase (RT) inhibitors. Further SAR studies and identification of a novel orally … G Campiani, F Aiello, M Fabbrini, E Morelli, A Ramunno, S Armaroli, ... Journal of medicinal chemistry 44 (3), 305-315, 2001 | 117 | 2001 |
| Synthesis, biological activity, and SARs of pyrrolobenzoxazepine derivatives, a new class of specific “peripheral-type” benzodiazepine receptor ligands G Campiani, V Nacci, I Fiorini, MP De Filippis, A Garofalo, SM Ciani, ... Journal of medicinal chemistry 39 (18), 3435-3450, 1996 | 114 | 1996 |
| Anxiolytic-like Effects of N,N-Dialkyl-2-phenylindol-3-ylglyoxylamides by Modulation of Translocator Protein Promoting Neurosteroid Biosynthesis F Da Settimo, F Simorini, S Taliani, C La Motta, AM Marini, S Salerno, ... Journal of medicinal chemistry 51 (18), 5798-5806, 2008 | 102 | 2008 |
| N,N-Dialkyl-2-phenylindol-3-ylglyoxylamides. A New Class of Potent and Selective Ligands at the Peripheral Benzodiazepine Receptor G Primofiore, F Da Settimo, S Taliani, F Simorini, MP Patrizi, E Novellino, ... Journal of medicinal chemistry 47 (7), 1852-1855, 2004 | 89 | 2004 |
| 3-Aryl[1,2,4]triazino[4,3-a]benzimidazol-4(10H)-ones: A New Class of Selective A1 Adenosine Receptor Antagonists F Da Settimo, G Primofiore, S Taliani, AM Marini, C La Motta, E Novellino, ... Journal of medicinal chemistry 44 (3), 316-327, 2001 | 72 | 2001 |
| Autosomal recessive familial exudative vitreoretinopathy: evidence for genetic heterogeneity G de Crecchio, F Simonelli, G Nunziata, S Mazzeo, GM Greco, E Rinaldi, ... Clinical genetics 54 (4), 315-320, 1998 | 72 | 1998 |
| Moderate hyperhomocysteinaemia and retinopathy in insulin-dependent diabetes O Vaccaro, D Ingrosso, A Rivellese, G Greco, G Riccardi The Lancet 349 (9058), 1102-1103, 1997 | 68 | 1997 |
| Derivatives of 4-Amino-6-hydroxy-2-mercaptopyrimidine as Novel, Potent, and Selective A3 Adenosine Receptor Antagonists B Cosimelli, G Greco, M Ehlardo, E Novellino, F Da Settimo, S Taliani, ... Journal of medicinal chemistry 51 (6), 1764-1770, 2008 | 67 | 2008 |
| Modeling of κ-opioid receptor/agonists interactions using pharmacophore-based and docking simulations A Lavecchia, G Greco, E Novellino, F Vittorio, G Ronsisvalle Journal of medicinal chemistry 43 (11), 2124-2134, 2000 | 66 | 2000 |
| New fluorescent 2-phenylindolglyoxylamide derivatives as probes targeting the peripheral-type benzodiazepine receptor: design, synthesis, and biological evaluation S Taliani, F Simorini, V Sergianni, C La Motta, F Da Settimo, B Cosimelli, ... Journal of Medicinal Chemistry 50 (2), 404-407, 2007 | 63 | 2007 |
| 2-(Benzimidazol-2-yl)quinoxalines: A Novel Class of Selective Antagonists at Human A1 and A3 Adenosine Receptors Designed by 3D Database Searching E Novellino, B Cosimelli, M Ehlardo, G Greco, M Iadanza, A Lavecchia, ... Journal of medicinal chemistry 48 (26), 8253-8260, 2005 | 63 | 2005 |
| Specific targeting highly conserved residues in the HIV-1 reverse transcriptase primer grip region. Design, synthesis, and biological evaluation of novel, potent, and broad … C Fattorusso, S Gemma, S Butini, P Huleatt, B Catalanotti, M Persico, ... Journal of medicinal chemistry 48 (23), 7153-7165, 2005 | 59 | 2005 |
| Use of comparative molecular field analysis and cluster analysis in series design E Novellino, C Fattorusso, G Greco Pharmaceutica Acta Helvetiae 70 (2), 149-154, 1995 | 59 | 1995 |
| Novel N2-Substituted Pyrazolo[3,4-d]pyrimidine Adenosine A3 Receptor Antagonists: Inhibition of A3-Mediated Human Glioblastoma Cell Proliferation S Taliani, C La Motta, L Mugnaini, F Simorini, S Salerno, AM Marini, ... Journal of medicinal chemistry 53 (10), 3954-3963, 2010 | 58 | 2010 |
