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Dr. Shankar Alegaon
Dr. Shankar Alegaon
KLE College of Pharmacy, KLE Academy of Higher Education and Research, Deemed to be University
E-mail confirmado em klepharm.edu
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Novel imidazo [2, 1-b][1, 3, 4] thiadiazole carrying rhodanine-3-acetic acid as potential antitubercular agents
SG Alegaon, KR Alagawadi, PV Sonkusare, SM Chaudhary, DH Dadwe, ...
Bioorganic & medicinal chemistry letters 22 (5), 1917-1921, 2012
1832012
Synthesis, characterization and antimicrobial activity evaluation of new 2, 4-Thiazolidinediones bearing imidazo [2, 1-b][1, 3, 4] thiadiazole moiety
KR Alagawadi, SG Alegaon
Arabian Journal of Chemistry 4 (4), 465-472, 2011
962011
1, 3, 4-Trisubstituted pyrazole analogues as promising anti-inflammatory agents
SG Alegaon, KR Alagawadi, MK Garg, K Dushyant, D Vinod
Bioorganic chemistry 54, 51-59, 2014
952014
New thiazolidinedione-5-acetic acid amide derivatives: synthesis, characterization and investigation of antimicrobial and cytotoxic properties
SG Alegaon, KR Alagawadi
Medicinal Chemistry Research 21, 816-824, 2012
542012
Synthesis of novel pyrazole–thiadiazole hybrid as potential potent and selective cyclooxygenase-2 (COX-2) inhibitors
SG Alegaon, MB Hirpara, KR Alagawadi, KK Hullatti, K Kashniyal
Bioorganic & Medicinal Chemistry Letters 24 (22), 5324-5329, 2014
502014
Synthesis, characterization and antimicrobial activity evaluation of new imidazo [2, 1-b][1, 3, 4] thiadiazole derivatives
SG Alegaon, KR Alagawadi
European Journal of Chemistry 2 (1), 94-99, 2011
372011
Three-component, one-pot synthesis of anthranilamide Schiff bases bearing 4-aminoquinoline moiety as Mycobacterium tuberculosis gyrase inhibitors
PS Salve, SG Alegaon, D Sriram
Bioorganic & medicinal chemistry letters 27 (8), 1859-1866, 2017
322017
New thiazolidine-2, 4-diones as antimicrobial and cytotoxic agent
SG Alegaon, KR Alagawadi
Medicinal Chemistry Research 21, 3214-3223, 2012
282012
Quinoline-azetidinone hybrids: Synthesis and in vitro antiproliferation activity against Hep G2 and Hep 3B human cell lines
SG Alegaon, P Parchure, LD Araujo, PS Salve, KR Alagawadi, ...
Bioorganic & Medicinal Chemistry Letters 27 (7), 1566-1571, 2017
232017
Synthesis, characterization, and biological evaluation of thiazolidine-2, 4-dione derivatives
SG Alegaon, KR Alagawadi, SM Pawar, D Vinod, U Rajput
Medicinal Chemistry Research 23, 987-994, 2014
212014
Synthesis and biological evaluation of 1, 3, 4-trisubstituted pyrazole analogues as anti-mycobacterial agents
SG Alegaon, MB Hirpara, KR Alagawadi, SS Jalalpure, VP Rasal, ...
Medicinal Chemistry Research 26, 1127-1138, 2017
162017
Synthesis and antitubercular activity of novel 3, 5-diaryl-4, 5-dihydro-1H-pyrazole derivatives
SG Alegaon, KR Alagawadi, DH Dadwe
Drug research, 553-558, 2014
162014
Synthesis of new 7-chloro-4-phenoxyquinoline analogues as potential antitubercular agents
PS Salve, SG Alegaon
Medicinal Chemistry Research 27 (1), 1-14, 2018
152018
Synthesis and biological evaluation of some 4-aminoquinoline derivatives as potential antitubercular agents
S Alegaon, K Kashniyal, S Kuncolienkar, R Kavalapure, P Salve, M Palled, ...
Future Journal of Pharmaceutical Sciences 6, 1-12, 2020
132020
Development and validation of UV-spectrophotometric method for determination of ciprofloxacin and curcumin in bulk powder
SS Sanjay, R Kavalapure, MS Palled, SG Alegaon
Int J Pharm Sci and Res 11, 1161-6, 2020
132020
Synthesis, antitubercular evaluation and docking studies of novel benzimidazole analogues
DML Araujo, MM Maste, S Alegaon, A Saxena
Int. J. Pharm. Sci. Res 9, 3696-3704, 2018
132018
Synthesis, pharmacophore modeling, and cytotoxic activity of 2-thioxothiazolidin-4-one derivatives
SG Alegaon, KR Alagawadi, D Vinod, B Unger, NA Khatib
Medicinal Chemistry Research 23, 5160-5173, 2014
132014
Synthesis, molecular docking and ADME studies of thiazole-thiazolidinedione hybrids as antimicrobial agents
SG Alegaon, V U, KR Alagawadi, D Kumar, RS Kavalapure, SD Ranade, ...
Journal of Biomolecular Structure and Dynamics 40 (14), 6211-6227, 2022
92022
Screening and assessment of selected alkaloids as potential inhibitors of COVID-19 protease enzyme.
SS Suryawanshi, RS Patil, PB Jayannache, MS Palled, SG Alegaon, ...
82020
Design, synthesis, and molecular docking study of some 2-((7-chloroquinolin-4-yl) amino) benzohydrazide Schiff bases as potential Eg5 inhibitory agents
RS Kavalapure, SG Alegaon, U Venkatasubramanian, AS Priya, ...
Bioorganic Chemistry 116, 105381, 2021
72021
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