| The emerging role of lysine methyltransferase SETD8 in human diseases C Milite, A Feoli, M Viviano, D Rescigno, A Cianciulli, AL Balzano, A Mai, ... Clinical epigenetics 8, 1-15, 2016 | 92 | 2016 |
| Discovery of a novel chemotype of histone lysine methyltransferase EHMT1/2 (GLP/G9a) inhibitors: rational design, synthesis, biological evaluation, and co-crystal structure C Milite, A Feoli, JR Horton, D Rescigno, A Cipriano, V Pisapia, M Viviano, ... Journal of medicinal chemistry 62 (5), 2666-2689, 2019 | 32 | 2019 |
| A continuous-flow synthesis of 1, 4-benzodiazepin-5-ones, privileged scaffolds for drug discovery M Viviano, C Milite, D Rescigno, S Castellano, G Sbardella RSC advances 5 (2), 1268-1273, 2015 | 27 | 2015 |
| Progress in the development of lysine methyltransferase SETD8 inhibitors C Milite, A Feoli, M Viviano, D Rescigno, A Mai, S Castellano, G Sbardella ChemMedChem 11 (16), 1680-1685, 2016 | 22 | 2016 |
| Turning nonselective inhibitors of type I protein arginine methyltransferases into potent and selective inhibitors of protein arginine methyltransferase 4 through a … G Iannelli, C Milite, N Marechal, V Cura, L Bonnefond, N Troffer-Charlier, ... Journal of Medicinal Chemistry 65 (17), 11574-11606, 2022 | 11 | 2022 |
| Pyrido oxazine derivatives as alk5 inhibitors P Daniele, D Pizzirani, P Bruno, M Biagetti, P Ronchi, S Guariento, ... US Patent App. 18/269,042, 2024 | | 2024 |
| Design, synthesis and biological evaluation of new small-molecule modulators of proein lysine methyltransferases (PKMTs) D Rescigno Universita degli studi di Salerno, 2018 | | 2018 |
| Design, synthesis and biological evaluation of new selective arginine methyltransferases (PRMTs) Inhibitors C Milite, A Feoli, D Rescigno, S Clarke, S Castellano, G Sbardella Italian-Spanish-Portuguese Joint Meeting in Medicinal Chemistry …, 2018 | | 2018 |
| Expanding the quinazoline ring to 3H-benzo [e][1, 4] diazepine: development of new and selective G9a inhibitors C Milite, A Feoli, D Rescigno, V Pisapia, S Cosconati, S Castellano, ... Italian-Spanish-Portuguese Joint Meeting in Medicinal Chemistry …, 2018 | | 2018 |
| Design, synthesis and biological evaluation of novel G9a inhibitors with improved brain permeability from a scaffold hopping approach D Rescigno, C Milite, M Viviano, A Feoli, S Castellano, G Sbardella Atti del XXVI Congresso Nazionale della Società Chimica Italiana, 67-67, 2017 | | 2017 |
| DESIGN, SYNTHESIS AND BIOLOGICAL EVALUATION OF NOVEL G9A INHIBITORS FROM A SCAFFOLD HOPPING APPROACH D Rescigno, C Milite, M Viviano, S Castellano, G Sbardella XXIV NMMC & 10th NPCF-September 11th-14th 2016, Perugia (Italy)-Book of …, 2016 | | 2016 |
| Identification of new inhibitors of PRMTs by a multi-substrate-adduct approach C Milite, D Rescigno, A Feoli, A Nunziata, S Castellano, G Sbardella XXIV NMMC & 10th NPCF-September 11th-14th 2016, Perugia (Italy)-Book of …, 2016 | | 2016 |
| A continuous-flow synthesis of 1, 4-benzodiazepin-5-ones, privileged scaffolds for drug discovery. D Rescigno, M Viviano, C Milite, G Sbardella, S Castellano XXIII National Meeting on Medicinal Chemistry (NMMC2015) and 9th Young …, 2015 | | 2015 |
