| Histone deacetylase inhibitor activity in royal jelly might facilitate caste switching in bees A Spannhoff, YK Kim, NJM Raynal, V Gharibyan, MB Su, YY Zhou, J Li, ... EMBO reports 12 (3), 238-243, 2011 | 220 | 2011 |
| Synthesis and Biochemical Evaluation of Δ2-Isoxazoline Derivatives as DNA Methyltransferase 1 Inhibitors S Castellano, D Kuck, M Viviano, J Yoo, F López-Vallejo, P Conti, ... Journal of medicinal chemistry 54 (21), 7663-7677, 2011 | 190 | 2011 |
| Arginine demethylation of G3BP1 promotes stress granule assembly WC Tsai, S Gayatri, LC Reineke, G Sbardella, MT Bedford, RE Lloyd Journal of Biological Chemistry 291 (43), 22671-22685, 2016 | 174 | 2016 |
| Epigenetic multiple ligands: mixed histone/protein methyltransferase, acetyltransferase, and class III deacetylase (sirtuin) inhibitors A Mai, D Cheng, MT Bedford, S Valente, A Nebbioso, A Perrone, ... Journal of medicinal chemistry 51 (7), 2279-2290, 2008 | 162 | 2008 |
| Dihydro(alkylthio)(naphthylmethyl)oxopyrimidines: Novel Non-Nucleoside Reverse Transcriptase Inhibitors of the S-DABO Series A Mai, M Artico, G Sbardella, S Quartarone, S Massa, AG Loi, A De Montis, ... Journal of Medicinal Chemistry 40 (10), 1447-1454, 1997 | 160 | 1997 |
| 5-Alkyl-2-(alkylthio)-6-(2,6-dihalophenylmethyl)-3,4-dihydropyrimidin-4(3H)-ones: Novel Potent and Selective Dihydro-alkoxy-benzyl-oxopyrimidine Derivatives A Mai, M Artico, G Sbardella, S Massa, E Novellino, G Greco, AG Loi, ... Journal of Medicinal Chemistry 42 (4), 619-627, 1999 | 159 | 1999 |
| Small-molecule inhibitors of histone acetyltransferase activity: identification and biological properties A Mai, D Rotili, D Tarantino, P Ornaghi, F Tosi, C Vicidomini, G Sbardella, ... Journal of medicinal chemistry 49 (23), 6897-6907, 2006 | 157 | 2006 |
| Structure-based design, synthesis, and biological evaluation of conformationally restricted novel 2-alkylthio-6-[1-(2, 6-difluorophenyl) alkyl]-3, 4-dihydro-5-alkylpyrimidin-4 … A Mai, G Sbardella, M Artico, R Ragno, S Massa, E Novellino, G Greco, ... Journal of medicinal chemistry 44 (16), 2544-2554, 2001 | 136 | 2001 |
| Preparation and anti-HIV-1 activity of Thio Analogues of Dichydroalkoxybenzyloxopyrimidines A Mai, M Artico, G Sbardella, S Massa, AG Loi, E Tramontano, P Scano, ... Journal of medicinal chemistry 38 (17), 3258-3263, 1995 | 135 | 1995 |
| Identification of long chain alkylidenemalonates as novel small molecule modulators of histone acetyltransferases G Sbardella, S Castellano, C Vicidomini, D Rotili, A Nebbioso, M Miceli, ... Bioorganic & medicinal chemistry letters 18 (9), 2788-2792, 2008 | 128 | 2008 |
| Small molecule inhibitors of histone arginine methyltransferases: homology modeling, molecular docking, binding mode analysis, and biological evaluations R Ragno, S Simeoni, S Castellano, C Vicidomini, A Mai, A Caroli, ... Journal of medicinal chemistry 50 (6), 1241-1253, 2007 | 126 | 2007 |
| Nε-lysine acetylation determines dissociation from GAP junctions and lateralization of connexin 43 in normal and dystrophic heart C Colussi, J Rosati, S Straino, F Spallotta, R Berni, D Stilli, S Rossi, ... Proceedings of the National Academy of Sciences 108 (7), 2795-2800, 2011 | 121 | 2011 |
| Constrained analogues of procaine as novel small molecule inhibitors of DNA methyltransferase-1 S Castellano, D Kuck, M Sala, E Novellino, F Lyko, G Sbardella Journal of medicinal chemistry 51 (7), 2321-2325, 2008 | 121 | 2008 |
| Computer-aided design, synthesis, and anti-HIV-1 activity in vitro of 2-alkylamino-6-[1-(2, 6-difluorophenyl) alkyl]-3, 4-dihydro-5-alkylpyrimidin-4 (3 H)-ones as novel potent … R Ragno, A Mai, G Sbardella, M Artico, S Massa, C Musiu, M Mura, ... Journal of medicinal chemistry 47 (4), 928-934, 2004 | 117 | 2004 |
| p300/CBP-associated factor selectively regulates the extinction of conditioned fear W Wei, CM Coelho, X Li, R Marek, S Yan, S Anderson, D Meyers, ... Journal of Neuroscience 32 (35), 11930-11941, 2012 | 102 | 2012 |
| 3-(4-Aroyl-1 H-pyrrol-2-yl)-N-hydroxy-2-propenamides, a new class of synthetic histone deacetylase inhibitors S Massa, A Mai, G Sbardella, M Esposito, R Ragno, P Loidl, G Brosch Journal of medicinal chemistry 44 (13), 2069-2072, 2001 | 102 | 2001 |
| Identification of 4-hydroxyquinolines inhibitors of p300/CBP histone acetyltransferases A Mai, D Rotili, D Tarantino, A Nebbioso, S Castellano, G Sbardella, ... Bioorganic & medicinal chemistry letters 19 (4), 1132-1135, 2009 | 97 | 2009 |
| The emerging role of lysine methyltransferase SETD8 in human diseases C Milite, A Feoli, M Viviano, D Rescigno, A Cianciulli, AL Balzano, A Mai, ... Clinical epigenetics 8, 1-15, 2016 | 91 | 2016 |
| Novel 3, 5-bis (bromohydroxybenzylidene) piperidin-4-ones as coactivator-associated arginine methyltransferase 1 inhibitors: enzyme selectivity and cellular activity D Cheng, S Valente, S Castellano, G Sbardella, R Di Santo, R Costi, ... Journal of medicinal chemistry 54 (13), 4928-4932, 2011 | 89 | 2011 |
| A New Facile and Expeditious Synthesis of N-Hydroxy-N′-Phenyloctanediamjde, a Potent Inducer of Terminal Cytodifferecntiation A Mai, M Esposito, G Sbardella, S Massa Organic Preparations and Procedures International 33 (4), 391-394, 2001 | 88 | 2001 |
Antonello MaiProfessore di Chimica Farmaceutica, Sapienza Università di RomaVerified email at uniroma1.it
