| Carborane clusters in computational drug design: a comparative docking evaluation using AutoDock, FlexX, Glide, and Surflex R Tiwari, K Mahasenan, R Pavlovicz, C Li, W Tjarks Journal of chemical information and modeling 49 (6), 1581-1589, 2009 | 109 | 2009 |
| Thiolates chemically induce redox activation of BTZ043 and related potent nitroaromatic anti-tuberculosis agents R Tiwari, GC Moraski, V Krchňák, PA Miller, M Colon-Martinez, ... Journal of the American Chemical Society 135 (9), 3539-3549, 2013 | 95 | 2013 |
| Virtually Complete Control of Simple and Face Diastereoselectivity in the Michael Addition Reactions between Achiral Equivalents of a Nucleophilic Glycine and (S)- or (R)-3 … VA Soloshonok, H Ueki, R Tiwari, C Cai, VJ Hruby The Journal of Organic Chemistry 69 (15), 4984-4990, 2004 | 90 | 2004 |
| Receptor-targeted liposomal delivery of boron-containing cholesterol mimics for boron neutron capture therapy (BNCT) BTS Thirumamagal, XB Zhao, AK Bandyopadhyaya, S Narayanasamy, ... Bioconjugate chemistry 17 (5), 1141-1150, 2006 | 79 | 2006 |
| Design, syntheses, and anti-TB activity of 1, 3-benzothiazinone azide and click chemistry products inspired by BTZ043 R Tiwari, PA Miller, LR Chiarelli, G Mori, M Šarkan, I Centárová, S Cho, ... ACS Medicinal Chemistry Letters 7 (3), 266-270, 2016 | 65 | 2016 |
| Syntheses and antituberculosis activity of 1, 3-benzothiazinone sulfoxide and sulfone derived from BTZ043 R Tiwari, PA Miller, S Cho, SG Franzblau, MJ Miller ACS medicinal chemistry letters 6 (2), 128-133, 2015 | 52 | 2015 |
| Electron delocalization in aminoguanidine: A computational study PV Bharatam, P Iqbal, A Malde, R Tiwari The Journal of Physical Chemistry A 108 (47), 10509-10517, 2004 | 51 | 2004 |
| Design and syntheses of anti-tuberculosis agents inspired by BTZ043 using a scaffold simplification strategy R Tiwari, U Möllmann, S Cho, SG Franzblau, PA Miller, MJ Miller ACS Medicinal Chemistry Letters 5 (5), 587-591, 2014 | 49 | 2014 |
| Carboranyl thymidine analogues for neutron capture therapy W Tjarks, R Tiwari, Y Byun, S Narayanasamy, RF Barth Chemical communications, 4978-4991, 2007 | 49 | 2007 |
| 3-Carboranyl thymidine analogues (3CTAs) and other boronated nucleosides for boron neutron capture therapy Y Byun, S Narayanasamy, J Johnsamuel, AK Bandyopadhyaya, R Tiwari, ... Anti-Cancer Agents in Medicinal Chemistry (Formerly Current Medicinal …, 2006 | 42 | 2006 |
| Hydrophilically enhanced 3-carboranyl thymidine analogues (3CTAs) for boron neutron capture therapy (BNCT) of cancer S Narayanasamy, BTS Thirumamagal, J Johnsamuel, Y Byun, ... Bioorganic & medicinal chemistry 14 (20), 6886-6899, 2006 | 38 | 2006 |
| Synthesis and evaluation of thymidine kinase 1-targeting carboranyl pyrimidine nucleoside analogs for boron neutron capture therapy of cancer HK Agarwal, A Khalil, K Ishita, W Yang, RJ Nakkula, LC Wu, T Ali, ... European journal of medicinal chemistry 100, 197-209, 2015 | 37 | 2015 |
| Synthesis, Biological Evaluation, and Radioiodination of Halogenated closo-Carboranylthymidine Analogues R Tiwari, A Toppino, HK Agarwal, T Huo, Y Byun, J Gallucci, ... Inorganic Chemistry 51 (1), 629-639, 2012 | 34 | 2012 |
| Application of (S)-and (R)-methyl pyroglutamates as inexpensive, yet highly efficient chiral auxiliaries in the asymmetric Michael addition reactions C Cai, T Yamada, R Tiwari, VJ Hruby, VA Soloshonok Tetrahedron letters 45 (37), 6855-6858, 2004 | 34 | 2004 |
| Synthesis and Biological Evaluation of Inhibitors of Thymidine Monophosphate Kinase from Bacillus Anthracis Y Byun, SR Vogel, AJ Phipps, C Carnrot, S Eriksson, R Tiwari, W Tjarks Nucleosides, Nucleotides and Nucleic Acids 27 (3), 244-260, 2008 | 23 | 2008 |
| Design, syntheses, and anti-tuberculosis activities of conjugates of piperazino-1, 3-benzothiazin-4-ones (pBTZs) with 2, 7-dimethylimidazo [1, 2-a] pyridine-3-carboxylic acids … MW Majewski, R Tiwari, PA Miller, S Cho, SG Franzblau, MJ Miller Bioorganic & medicinal chemistry letters 26 (8), 2068-2071, 2016 | 15 | 2016 |
| Michael addition reactions between various nucleophilic glycine equivalents and (S, E)-1-enoyl-5-oxo-N-phenylpyrrolidine-2-carboxamide, an optimal type of chiral Michael … TK Ellis, H Ueki, R Tiwari, VA Soloshonok Tetrahedron: Asymmetry 20 (22), 2629-2634, 2009 | 13 | 2009 |
| Comparative molecular field analysis and comparative molecular similarity indices analysis of boron-containing human thymidine kinase 1 substrates AK Bandyopadhyaya, R Tiwari, W Tjarks Bioorganic & medicinal chemistry 14 (20), 6924-6932, 2006 | 13 | 2006 |
| Boron cluster (radio) halogenation in biomedical research HK Agarwal, S Hasabelnaby, R Tiwari, W Tjarks Boron Science: New Technologies and Applications, 108-144, 2011 | 12 | 2011 |
| Cellular influx, efflux, and anabolism of 3-carboranyl thymidine analogs: potential boron delivery agents for neutron capture therapy E Sjuvarsson, VL Damaraju, D Mowles, MB Sawyer, R Tiwari, HK Agarwal, ... Journal of Pharmacology and Experimental Therapeutics 347 (2), 388-397, 2013 | 11 | 2013 |
Rolf F BarthProfessor of Pathology, The Ohio State UniversityE-mail confirmado em osumc.edu
